With Heterocyclic Compound Patents (Class 514/66)
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Publication number: 20130338002Abstract: Disclosed are compounds of Formula 1, wherein X is O or S; Y is O or S; and R1, R2, R3 and R4 are as defined in the disclosure. Also disclosed are compositions containing the compounds of Formula 1 and methods for controlling an invertebrate pest comprising contacting the invertebrate pest or its environment with a biologically effective amount of a compound or a composition of the invention.Type: ApplicationFiled: August 15, 2013Publication date: December 19, 2013Applicant: E I DU PONT DE NEMOURS AND COMPANYInventors: CALEB WILLIAM HOLYOKE, JR., WENWING ZHANG
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Publication number: 20130261083Abstract: The invention relates to additives enhancing the activity of certain insecticides, to significantly increase the effect of such insecticides when applied to the exterior foliage of a plant, thus increasing the kill rate of feeding insects that are normally protected deep within other tissue structures of the plant.Type: ApplicationFiled: December 9, 2011Publication date: October 3, 2013Applicant: Akzo Nobel Chemicals International B.V.Inventors: James Lyle Hazen, Jinxia Susan Sun
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Publication number: 20130143829Abstract: The present invention provides pyrethroid/macrocyclic lactone-containing topical formulations that are effective against animal pests, including ecto- and endoparasites. The formulations may be used for combating parasites in or on birds and mammals. The invention also provides for an improved method for eradicating, controlling and preventing parasite and/or pest infestation of birds and mammals.Type: ApplicationFiled: December 6, 2011Publication date: June 6, 2013Inventor: Robert Holmes
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Patent number: 8404649Abstract: This invention recites naphthyl isoxazoline oxime derivatives of Formula (1) geometric isomers, stereoisomers thereof, pharmaceutically or veterinarily acceptable salts thereof, compositions thereof, and their use as a parasiticide in animals. The variables, R1a, R1b, R1c, R2, R3, and are as described herein.Type: GrantFiled: September 15, 2011Date of Patent: March 26, 2013Assignee: AH USA 42 LLCInventors: Michael Curtis, Edmund L. Ellsworth
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Publication number: 20120245126Abstract: Nitromethylene analogues of imidacloprid and divalent and oxabridged heterocyclic neonicotinoid compounds constructed by dialdehydes, preparation methods and uses thereof are disclosed. Compounds represented by formula (A) or (B), their optical isomers or agrochemically acceptable salts are provided. Agrochemical compositions comprising the said compounds, their optical isomers or agrochemically acceptable salts, the uses of the said agrochemical compositions and the preparation methods of the said compounds, their optical isomers or agrochemically acceptable salts are also disclosed. The compounds and their derivatives have high insecticidal activities to several farming and forestry pests including homoptera and lepidoptera pests, such as aphis, fulgorid, whitefly, leafhopper, common thrips, cotton bollworm, cabbage caterpillar, cabbage moth, cotton leafworm and armyworm.Type: ApplicationFiled: December 9, 2010Publication date: September 27, 2012Applicant: EAST CHINA UNIVERSITY OF SCIENCE AND TECHNOLOGYInventors: Xuhong Qian, Zhong Li, Xusheng Shao, Xiaoyong Xu, Zhiping Xu, Gonghua Song
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Publication number: 20120171127Abstract: Certain surfactants suitable for use alone to dissolve a water-insoluble component in compositions is described for providing VOC-free compressed gas aerosol compositions. The compositions include water-insoluble component(s), a surfactant and water. The water-insoluble component(s) can be active agent(s), such as fragrance(s) and/or an insecticide(s). The surfactant is present as a single surfactant which, in the absence of a solvent, dissolves or disperses the water-insoluble component(s) and provides a homogenous blend in water which provides a stable compressed gas emulsion.Type: ApplicationFiled: March 12, 2012Publication date: July 5, 2012Applicant: S.C. JOHNSON & SON, INC.Inventors: Richard S. VALPEY, III, Paul A. CLARK, Jessica A. HEISER
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Patent number: 8178122Abstract: Materials and methods, for preparation of coatings based on titanium dioxide for osteointegrated biomedical prostheses. The coatings may comprise nanomaterials having antibacterial properties. For example, an endo-osseous implant is provided with a coating comprised of nanocrystalline material comprising nanoparticles of formula (I) (L-Men+)i,??(I) where AOx represents TiO2 or ZrO2; Men+ is a metallic ion having antibacterial activity, with n=1 or 2; L is a bi functional organic molecule which can simultaneously bind to the metal oxide and to the metallic ion Men+, and i is the number of L-Men+ groups bound to one nanoparticle of AOx.Type: GrantFiled: August 14, 2006Date of Patent: May 15, 2012Assignee: NM Tech Nanomaterials and Microdevices Technology Ltd.Inventors: Carlo Alberto Bignozzi, Francesco Carinci, Stefano Caramori, Valeria Dissette
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Patent number: 8158137Abstract: The present invention relates to nanomaterials comprised of metal oxides associated with cationic metals having antibacterial activity. In particular, the present invention relates to nanocrystalline compounds of formula (I): AOx-(L-Men+) i, (I) where AOx represents the metal oxide or metalloid oxide, with x=1 or 2; Me11“1” is a metal ion having antibacterial activity, with n=1 or 2; L is a bifunctional molecule, either organic or organometallic, capable of binding simultaneously with the metal oxide or metalloid oxide and the metal ion Men+; and i represents the number of L-Men+groups bound to a AOx nanoparticle.Type: GrantFiled: April 24, 2006Date of Patent: April 17, 2012Assignee: NM Tech Nanomaterials and Microdevices Technology LimitedInventors: Carlo Alberto Bignozzi, Valeria Dissette, Alfredo Corallini, Giacomo Carra′, Renato Della Valle
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Publication number: 20120077765Abstract: This invention recites naphthyl isoxazoline oxime derivatives of Formula (1) geometric isomers, stereoisomers thereof, pharmaceutically or veterinarily acceptable salts thereof, compositions thereof, and their use as a parasiticide in animals. The variables, R1a, R1b, R1c, R2, R3, and are as described herein.Type: ApplicationFiled: September 15, 2011Publication date: March 29, 2012Applicant: PFIZER INC.Inventors: Michael Curtis, Edmund L. Ellsworth
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Publication number: 20120058974Abstract: The present invention relates to an agrochemical composition comprising pesticide and UV absorber. The invention furthermore relates to UV-absorbers and to the use thereof in agrochemical compositions. It moreover relates to a method of controlling phytopathogenic fungi and/or undesirable plant growth and/or undesirable insect or mite infestation and/or of regulating plant growth.Type: ApplicationFiled: March 10, 2010Publication date: March 8, 2012Applicant: BASF SEInventors: Andrea Misske, Christian Bittner, Michael Ishaque, Markus Hoffmann, Richard Riggs, Ruediger Sens, Andre Kabat, Sylke Haremza, Douglas D. Anspaugh, David M. Terry
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Patent number: 8097603Abstract: The present invention relates to novel skin-friendly dermally applicable liquid formulations comprising a pyrethrin or pyrethroid and MGK 264 in a ratio of at least 1:20 and a further insecticide, preferably from the group of the neonicotinoids, for controlling parasitic arthropods on animals.Type: GrantFiled: April 24, 2004Date of Patent: January 17, 2012Assignee: Bayer Animal Health GmbHInventors: Kirkor Sirinyan, Andreas Turberg
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Patent number: 7612093Abstract: Provided are methods and compositions for treating hepatitis virus infections in mammals, especially humans. The methods comprise (1) administering N-substituted-1,5-dideoxy-1,5-imino-D-glucitol compounds in combination with nucleoside antiviral agents, nucleotide antiviral agents, mixtures thereof, or immunomodulating/immunostimulating agents, or (2) administering N-substituted-1,5-dideoxy-1,5-imino-D-glucitol compounds in combination with nucleoside antiviral agents, nucleotide antiviral agents, or mixtures thereof, and immunomodulating/immunostimulating agents.Type: GrantFiled: December 15, 2005Date of Patent: November 3, 2009Assignee: United Therapeutics CorporationInventors: Gary S. Jacob, Timothy M. Block, Raymond A. Dwek
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Publication number: 20080287294Abstract: A method of controlling mollusc damage to plants in horticulture or agriculture comprises treating the plant's propagation material with a combination comprising (I) one or more of (i) one or more of a neonicotinoid, (ii) one or more of a pyrethroid, (iii) one or more of a macrolide, and (iv) one or more of a defined bisamide compound, and (II) one or more of metaldehyde, methiocarb, thiodicarb, cinnamaldehyde and 3,5, dimethoxycinnamic acid, and optionally one or more customary formulation auxiliaries.Type: ApplicationFiled: April 6, 2006Publication date: November 20, 2008Applicant: SYNGENTA CROP PROTECTION, INC.Inventors: Martin Weiss, Franz Brandl
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Publication number: 20080090780Abstract: A storage stable, efficacious pesticide formulation is provided that is dilutable by the user and contains azadirachtin (AZA) and a pyrethrin or pyrethroid (PYR), and optionally an aprotic solvent and non-ionic, substantially water-free emulsifier. A sufficient amount of the PYR is provided to complex with the AZA A on opposite sides of the molecular structure thereof, thereby preventing rearrangement of the AZA A molecule in the presence of moisture that would result in hydrolysis and decomposition of AZA A. The AZA-PYR combination is sufficiently chemically stable such that less than 10% of the AZA A is decomposed when the formulation is subjected to an accelerated aging test for 30 days at 40° C. in a sealed container. The molar ratio of PYR to AZA A is preferably within the range of 0.5/1-10.5/1, more preferably within the range of 1.5/1-7/1, and most preferably with the range of 3/1-6/1.Type: ApplicationFiled: October 13, 2006Publication date: April 17, 2008Applicant: PBI/GORDON CORPORATIONInventors: Dale R. Sanson, James A. Armbruster
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Publication number: 20040077602Abstract: The present invention relates to a mixture composition for controlling ectoparasites of mammals and birds, comprising as active ingredients a compound of formula (I) or a salt thereof and one or more compounds selected from the group consisting of pyrethroid insecticides. The composition according to the present invention has high control effect against resistant ectoparasites, can quickly act, and is safe.Type: ApplicationFiled: October 9, 2003Publication date: April 22, 2004Applicant: Meiji Seika Kaisha, Ltd.Inventor: Kazuhiko Oyama
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Publication number: 20030166618Abstract: Composition for controlling insects and representatives of the order Acarina, which comprises a combination of variable amounts of one or more compounds of the formula 1Type: ApplicationFiled: February 4, 2003Publication date: September 4, 2003Inventors: Robert Senn, Peter Maienfisch, Peter Wyss
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Publication number: 20030161896Abstract: Novel active compound combinations of compounds of the formula (I) 1Type: ApplicationFiled: February 21, 2003Publication date: August 28, 2003Inventors: Astrid Mauler-Machnik, Ulrike Wachendorff-Neumann, Herbert Gayer
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Publication number: 20030148999Abstract: The novel active compound combinations of certain cyclic ketoenols and the active compounds (1) to (23) listed in the description have very good insecticidal and acaricidal properties.Type: ApplicationFiled: December 19, 2002Publication date: August 7, 2003Inventors: Reiner Fischer, Christoph Erdelen
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Patent number: 6518274Abstract: The invention relates to the use of cycloventabenzofuran derivatives for the production of a medicament for the treatment of nuclear factor of &kgr;B-dependent diseases.Type: GrantFiled: April 18, 2001Date of Patent: February 11, 2003Assignee: Bayer AktiengesellschaftInventors: Matthias Gehling, Jörg Baumgarten, Axel Kretschmer, Horst-Peter Antonicek, Peter Proksch, Bambang Wahyu Nugroho, Frank Bohnenstengel
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Patent number: 6506396Abstract: A stable medicated animal care formulation including, by weight; (a) 0.1-10% of an active agricultural ingredient, of an animal care and/or veterinary reagents, (b) 0.0002-40% of a microemulsion concentrate including: (i) 0-10% of a castor oil ethoxylate or tristyryl phenol ethoxylate, (ii) 0-1% of an ethoxylated phosphoric acid as pH buffer, (iii) 0.0002-4% of a N—C8-C18 alkyl pyrrolidone and (iv) 0-6% of a N—C1-C4 alkyl pyrrolidone, (c) a surfactant with shampoo properties, and (d) water, wherein (c)+(d) is 50-99.4%.Type: GrantFiled: September 6, 2001Date of Patent: January 14, 2003Assignee: ISP Investments Inc.Inventors: Kolazi S. Narayanan, Domingo I. Jon, Donald I. Prettypaul
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Patent number: 6355609Abstract: Nutritional solutions and methods of making same are disclosed. The solutions include protein, lipid, and a carbohydrate source including high amylose starch and guar gum.Type: GrantFiled: April 14, 1999Date of Patent: March 12, 2002Assignee: Nestec S.A.Inventors: Chandrasekhara Reddy Mallangi, Eileen Fuchs, Kjerstin Carlsson, Axel Syrbe, Reinhard Behringer
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Publication number: 20020010142Abstract: A parasiticidal formulation is provided. This formulation includes a pyrrolidone solvent, a bridging solvent, and an parasiticidal agent. One or more parasiticidal agents may be included in the formulation. Preferably, the formulation contains both closantel and ivermectin. Another aspect of the present invention is a method of making this parasiticidal formulation. This method includes mixing a pyrrolidone solvent and a bridging solvent to form a solvent solution and adding one or more parasiticidal agents to the solvent solution. A further aspect of the present invention is a method for administering the parasiticidal formulation of the present invention to an animal. This method of administration includes providing the parasiticidal formulation described above and applying this formulation to the skin of an animal, wherein the formulation is absorbed through the animal's skin.Type: ApplicationFiled: September 26, 2001Publication date: January 24, 2002Inventor: Richard Mihalik
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Patent number: 6045816Abstract: A clear, one-phase, efficacious aqueous microemulsion of an agriculturally active pyrethroid insecticide for delivery at a high loading of active is provided herein which is free of nonylphenol ethoxylate.Type: GrantFiled: June 17, 1998Date of Patent: April 4, 2000Assignee: ISP Investments Inc.Inventors: Kolazi S. Narayanan, Domingo Jon, Robert M. Ianniello, Donald Prettypaul
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Patent number: 5679662Abstract: In an insecticidal formulation containing Pyrethrum, addition of appropriate amounts of azadirachtin and clarified neem oil can significantly synergize the Pyrethrum activity while reducing or eliminating the need for Pipronyl butoxide as an agent to augment Pyrethrum activity. The disclosed formulations represent a significant cost advantage when compared to existing Pyrethrum/Pipronyl butoxide formulations.Type: GrantFiled: June 6, 1995Date of Patent: October 21, 1997Assignee: Thermo Trilogy CorporationInventors: Pauley Fei-Zan Chang, James F. Walter, Jerrold R. Harris
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Patent number: 5591727Abstract: The invention relates to an insecticidal composition which comprises at least one pyrethroid, at least one UV absorbing agent and at least one antioxidant from the group consisting of tocopherol derivatives and citric acid esters. This insecticidal composition can in particular be used as an emulsion or on a powdery carrier for the control of flying and crawling insects such as flies and cockroaches.Type: GrantFiled: February 7, 1995Date of Patent: January 7, 1997Assignees: Perycut-Chemie AG, Franz BencsitsInventor: Franz Bencsits
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Patent number: 5407920Abstract: A method of treating wood and timber is disclosed. Wood or timber is treated with a pesticidal microemulsion or other water-miscible formulation that has an average particle size of at most 200 nm. The treatment is particularly effective in protecting wood and timber against the common furniture beetle (Anobium punctatum), the house longhorn (Hylotrupes bajulus), the death watch beetle (Xestobium rufovillorum), dry rot (Serpula (merulius) lacrymans) and wet rot (Coniophora puteena).Type: GrantFiled: August 26, 1993Date of Patent: April 18, 1995Assignee: NC Development, Inc.Inventor: Howard B. Dawson
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Patent number: 5242907Abstract: Tropical and temperate crops, particularly rice, maize, cotton, soya and fruit, can be protected, particularly against insect pests of the orders Leoidoptera, Diptera, Coleoptera, Hemiptera, Orthoptera, Dictyoptera, Hymenoptera and Isoctera and acarine pests, by treatment with a pesticidal water-miscible formulation whose average particle size is at most 200 nm. Public health pests, including the house fly (Musca domestica), cockroach (Blatta sp. or Periplaneta sp.) and mosquito (Aedes aegyoti) as well as pests which infest or affect timber, particularly in buildings, can also be controlled with such formulations. The formulations include water, oil, a surfactant, and a cosurfactant, wherein either the oil is a pesticide or the formulation comprises a pesticide dissolved in the oil. The pesticide may be a pyrethroid such as cypermethrin or deltamethrin. The formulations can be molecular solutions, micellar solutions or microemulsions (water-in-oil or oil-in-water) and are generally clear.Type: GrantFiled: April 29, 1991Date of Patent: September 7, 1993Assignee: NC Development, Inc.Inventor: Howard B. Dawson
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Patent number: 5017563Abstract: Castanospermine mono- and di-esters and glycosides active as inhibitors of carbohydrate digestive enzymes and useful in treating diabetes are described herein. The compounds are prepared by the reaction of castanospermine with an appropriate acid halide or anhydride or with an appropriate glycosyl halide or glycosyl acetimidate under conditions which would favor the isolation of the mono- and di-esterified and glycosylated products. Various blocking groups, which can be selectively removed under mild conditions, can also be used to favor the formation of certain isomers.Type: GrantFiled: May 1, 1990Date of Patent: May 21, 1991Assignee: Merrell Dow Pharmaceuticals Inc.Inventors: Paul S. Liu, Barry L. Rhinehart, John K. Daniel
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Patent number: 4983591Abstract: A combination of pyrethrum and fatty acid salt materials has been formulated which produces a stable, commercially useful, and environmentally safe pesticide. The specific composition comprises an aqueous solution having a pH within the range of 7.5 to 8.8; an aqueous solution comprising at least about 0.5 percent by weight of monocarboxylic acids and their alkali metal salts, where the acid mixture is at least 70% oleic acid and 6% linoleic acid; a pyrethrum extract; a solvent for the pyrethrum, which is preferably a 2-6 carbon alcohol; a trace amount of an antioxidant. The composition is effective against insects of at least the orders Homoptera, Coleoptera, Dermaptera, Hemiptera, and Lepidoptera, and against crustacea of the order Isopoda.Type: GrantFiled: November 6, 1989Date of Patent: January 8, 1991Assignee: Safer, Ltd.Inventors: George S. Puritch, Gregory S. Salloum, Willem W. Nijholt
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Patent number: 4956353Abstract: Kojic acid and its esters have been found to be more effective synergists for pyrethroid and carbamate insecticides on H. zea and S. frugiperda. Thus they may serve as replacements for the widely used methylene dioxyphenyl compounds such as piperonyl butoxide.Type: GrantFiled: June 16, 1988Date of Patent: September 11, 1990Assignee: The United States of America as represented by the Secretary of AgricultureInventor: Patrick F. Dowd
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Patent number: 4904645Abstract: A combination of pyrethrum and fatty acid salt materials has been formulated which produces a stable, commercially useful, and environmentally safe pesticide. The specific composition comprises an aqueous solutioon having a pH within the range of 7.5 to 8.8; an aqueous solution comprising about 50% by weight of monocarboxylic acids and their alkali metal salts, where the acid mixture is at least 70% oleic acid and 6% linoleic acid; a pyrethrum extract; a solvent for the pyrethrum, which is preferably a 2-6 carbon alcohol; a trace amount of an antioxidant. The composition is effective against insects of at least the orders Homoptera, Coleoptera, Dermaptera, Hemiptera, and Lepidoptera, and against crustacea of the order Isopoda.Type: GrantFiled: January 27, 1988Date of Patent: February 27, 1990Assignee: Safer, Ltd.Inventors: George S. Puritch, Gregory S. Salloum, Willem W. Nijholt
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Patent number: 4569928Abstract: Novel esters in all possible isomeric forms and mixtures thereof of the formula ##STR1## wherein R is selected from the group consisting of (a) optionally unsaturated alkyl of 1 to 18 carbon atoms and optionally unsaturated cycloalkyl or cycloalkylalkyl of 3 to 8 carbon atoms optionally substituted with at least one member of the group consisting of halogen, --OH, --SH, --OR', --SR', --NO.sub.2, ##STR2## --SO.sub.2 AlK.sub.2, --SO.sub.3 AlK.sub.3, aryl optionally substituted with at least one member of the group consisting of --OH, alkoxy of 1 to 8 carbon atoms, alkyl of 1 to 8 carbon atoms, halogen, --CF.sub.3, --OCF.sub.3, --SCF.sub.3 and ##STR3## R' is alkyl of 1 to 8 carbon atoms, R" and R'" are individually selected from the group consisting of hydrogen and alkyl of 1 to 8 carbon atoms, AlK.sub.1, AlK.sub.2 and AlK.sub.Type: GrantFiled: October 28, 1983Date of Patent: February 11, 1986Assignee: Roussel UclafInventors: Jean Tessier, Andre Teche, Jean-Pierre Demoute